id	sid	eid	entity	type
admet-530	1	1	10.5599	CARDINAL
admet-530	1	2	74	CARDINAL
admet-530	1	3	admet &	ORG
admet-530	1	4	6(2	CARDINAL
admet-530	1	5	2018	DATE
admet-530	1	6	74	CARDINAL
admet-530	1	7	issn	PERSON
admet-530	1	8	1848-7718	DATE
admet-530	1	9	discovery	PRODUCT
admet-530	1	10	robert j. young* drug	PERSON
admet-530	1	11	glaxosmithkline medicines research centre	ORG
admet-530	1	12	stevenage	GPE
admet-530	1	13	sg1 2ny	DATE
admet-530	1	14	uk	GPE
admet-530	1	15	rob.j.young@gsk.com	ORG
admet-530	2	1	+44 1738 551372	ORG
admet-530	2	2	march 29, 2018	DATE
admet-530	2	3	may 16, 2018	DATE
admet-530	2	4	may 25, 2018	DATE
admet-530	2	5	discovery	PRODUCT
admet-530	4	1	100	CARDINAL
admet-530	6	1	1,2	CARDINAL
admet-530	7	1	2,3	CARDINAL
admet-530	7	2	4,5	CARDINAL
admet-530	9	1	6	CARDINAL
admet-530	10	1	6	CARDINAL
admet-530	12	1	the past decade	DATE
admet-530	13	1	6(2	CARDINAL
admet-530	13	2	2018	DATE
admet-530	13	3	74	CARDINAL
admet-530	13	4	10.5599	CARDINAL
admet-530	13	5	75	CARDINAL
admet-530	13	6	8	CARDINAL
admet-530	15	1	9	CARDINAL
admet-530	15	2	10	CARDINAL
admet-530	16	1	adme	ORG
admet-530	17	1	11	CARDINAL
admet-530	18	1	12	CARDINAL
admet-530	18	2	hsa	ORG
admet-530	20	1	13	CARDINAL
admet-530	23	1	8	CARDINAL
admet-530	24	1	1	CARDINAL
admet-530	25	1	10 mm	QUANTITY
admet-530	26	1	50	CARDINAL
admet-530	26	2	l	NORP
admet-530	26	3	96	CARDINAL
admet-530	27	1	5l	CARDINAL
admet-530	27	2	50/50	CARDINAL
admet-530	32	1	2	CARDINAL
admet-530	38	1	s. bunnally	PERSON
admet-530	38	2	r.j. young admet &	ORG
admet-530	38	3	6(2	CARDINAL
admet-530	38	4	2018	DATE
admet-530	38	5	74	CARDINAL
admet-530	38	6	1	CARDINAL
admet-530	39	1	100	CARDINAL
admet-530	39	2	weekly	DATE
admet-530	40	1	first	ORDINAL
admet-530	40	2	14	CARDINAL
admet-530	42	1	15	CARDINAL
admet-530	44	1	50 x 2 mm	QUANTITY
admet-530	44	2	uk	GPE
admet-530	44	3	7.4	CARDINAL
admet-530	44	4	10.5	CARDINAL
admet-530	45	1	9	CARDINAL
admet-530	46	1	1	CARDINAL
admet-530	47	1	10	CARDINAL
admet-530	48	1	two	CARDINAL
admet-530	49	1	3	CARDINAL
admet-530	49	2	3	CARDINAL
admet-530	50	1	3	CARDINAL
admet-530	50	2	log p	ORG
admet-530	50	3	non-zwitterionic	ORG
admet-530	51	1	0.0857)*chi 2.00	CARDINAL
admet-530	52	1	1	CARDINAL
admet-530	52	2	6(2	CARDINAL
admet-530	52	3	2018	DATE
admet-530	52	4	74	CARDINAL
admet-530	52	5	10.5599	CARDINAL
admet-530	52	6	77	CARDINAL
admet-530	52	7	2	CARDINAL
admet-530	53	1	2	CARDINAL
admet-530	53	2	7.4 x x x x	QUANTITY
admet-530	53	3	10.5	CARDINAL
admet-530	54	1	3	CARDINAL
admet-530	54	2	7.4	CARDINAL
admet-530	55	1	1,10	CARDINAL
admet-530	55	2	discovery	PRODUCT
admet-530	56	1	2,18	CARDINAL
admet-530	57	1	19	CARDINAL
admet-530	57	2	lle =	PERSON
admet-530	58	1	20	CARDINAL
admet-530	59	1	21	CARDINAL
admet-530	60	1	22,23	CARDINAL
admet-530	61	1	d7.4 + #	FAC
admet-530	61	2	13	CARDINAL
admet-530	61	3	6	CARDINAL
admet-530	61	4	100	CARDINAL
admet-530	61	5	g	ORG
admet-530	62	1	s. bunnally	PERSON
admet-530	62	2	r.j. young admet &	ORG
admet-530	62	3	6(2	CARDINAL
admet-530	62	4	2018	DATE
admet-530	62	5	74	CARDINAL
admet-530	62	6	hsa	ORG
admet-530	62	7	50	CARDINAL
admet-530	62	8	3 mm	QUANTITY
admet-530	62	9	france	GPE
admet-530	62	10	up to 30 %	PERCENT
admet-530	62	11	50 mm	QUANTITY
admet-530	62	12	7.4	CARDINAL
admet-530	63	1	24	CARDINAL
admet-530	65	1	hsa	ORG
admet-530	66	1	hsa	ORG
admet-530	66	2	2	CARDINAL
admet-530	68	1	2	CARDINAL
admet-530	69	1	4	CARDINAL
admet-530	70	1	hsa	ORG
admet-530	70	2	hplc measurement	ORG
admet-530	70	3	3	CARDINAL
admet-530	72	1	hsa	ORG
admet-530	74	1	hsa	ORG
admet-530	74	2	hsa	ORG
admet-530	74	3	4a	CARDINAL
admet-530	74	4	6(2	CARDINAL
admet-530	74	5	2018	DATE
admet-530	74	6	74	CARDINAL
admet-530	74	7	10.5599	CARDINAL
admet-530	74	8	79	CARDINAL
admet-530	75	1	hsa	ORG
admet-530	75	2	4b	CARDINAL
admet-530	77	1	25	CARDINAL
admet-530	77	2	100	CARDINAL
admet-530	77	3	4.6	CARDINAL
admet-530	77	4	10	CARDINAL
admet-530	77	5	regis	ORG
admet-530	77	6	west lafayette	GPE
admet-530	78	1	26	CARDINAL
admet-530	79	1	up to 85 %	PERCENT
admet-530	80	1	kiam	PERSON
admet-530	82	1	0.046*chiiam	CARDINAL
admet-530	85	1	chiiam	PERSON
admet-530	85	2	27	CARDINAL
admet-530	85	3	28	CARDINAL
admet-530	85	4	29	CARDINAL
admet-530	87	1	iam	ORG
admet-530	87	2	hsa	ORG
admet-530	87	3	5	CARDINAL
admet-530	88	1	5	CARDINAL
admet-530	89	1	iam	ORG
admet-530	89	2	hplc measurement	ORG
admet-530	89	3	kiam =	PERSON
admet-530	90	1	0.046*chiiam	CARDINAL
admet-530	92	1	hplc demax drug	ORG
admet-530	92	2	3	CARDINAL
admet-530	93	1	30	CARDINAL
admet-530	94	1	4	CARDINAL
admet-530	95	1	31	CARDINAL
admet-530	95	2	hsa	ORG
admet-530	95	3	iam	ORG
admet-530	95	4	6	CARDINAL
admet-530	96	1	32	CARDINAL
admet-530	96	2	hsa	ORG
admet-530	96	3	iam	ORG
admet-530	96	4	33	CARDINAL
admet-530	97	1	34	CARDINAL
admet-530	98	1	r.j. young admet &	ORG
admet-530	98	2	6(2	CARDINAL
admet-530	98	3	2018	DATE
admet-530	98	4	74	CARDINAL
admet-530	98	5	hplc demax	ORG
admet-530	98	6	7	CARDINAL
admet-530	98	7	7	CARDINAL
admet-530	99	1	1 %	PERCENT
admet-530	101	1	biophaseconc (	ORG
admet-530	102	1	3	CARDINAL
admet-530	102	2	2	CARDINAL
admet-530	102	3	0.23	CARDINAL
admet-530	102	4	kiam -0.72	PERSON
admet-530	102	5	4	CARDINAL
admet-530	102	6	max	PERSON
admet-530	102	7	100 %	PERCENT
admet-530	105	1	6	CARDINAL
admet-530	107	1	29	CARDINAL
admet-530	107	2	log10	PERSON
admet-530	108	1	8	CARDINAL
admet-530	108	2	d7.4	WORK_OF_ART
admet-530	111	1	6(2	CARDINAL
admet-530	111	2	2018	DATE
admet-530	111	3	74	CARDINAL
admet-530	111	4	10.5599	CARDINAL
admet-530	111	5	81	CARDINAL
admet-530	111	6	first	ORDINAL
admet-530	112	1	7	CARDINAL
admet-530	113	1	8	CARDINAL
admet-530	114	1	6	CARDINAL
admet-530	114	2	2	CARDINAL
admet-530	114	3	r.j. young admet &	ORG
admet-530	114	4	6(2	CARDINAL
admet-530	114	5	2018	DATE
admet-530	114	6	74	CARDINAL
admet-530	116	1	hsa	ORG
admet-530	116	2	iam	ORG
admet-530	118	1	gsk phys chem group	ORG
admet-530	118	2	klara valko	PERSON
admet-530	118	3	alan hill	PERSON
admet-530	119	1	1	CARDINAL
admet-530	119	2	n.a. meanwell	ORG
admet-530	119	3	ed	PERSON
admet-530	119	4	springer berlin heidelberg	GPE
admet-530	119	5	berlin	GPE
admet-530	119	6	heidelberg	GPE
admet-530	119	7	2014	DATE
admet-530	120	1	1-68	CARDINAL
admet-530	121	1	2	CARDINAL
admet-530	123	1	24 (2011	DATE
admet-530	123	2	1420	CARDINAL
admet-530	124	1	3	CARDINAL
admet-530	124	2	gleeson	PERSON
admet-530	124	3	p.d. leeson	PERSON
admet-530	124	4	der waterbeemd	PERSON
admet-530	124	5	chapter 1	LAW
admet-530	125	1	1-31	DATE
admet-530	126	1	4	CARDINAL
admet-530	126	2	leeson	PERSON
admet-530	126	3	b. springthorpe	PERSON
admet-530	128	1	nat rev drug discov	PERSON
admet-530	128	2	6 (2007	DATE
admet-530	128	3	881	CARDINAL
admet-530	129	1	5	CARDINAL
admet-530	129	2	leeson	PERSON
admet-530	129	3	r.j.	PERSON
admet-530	131	1	6	CARDINAL
admet-530	131	2	722	CARDINAL
admet-530	132	1	6	CARDINAL
admet-530	132	2	m.p. gleeson	PERSON
admet-530	132	3	a. hersey	PERSON
admet-530	132	4	d. montanari	PERSON
admet-530	132	5	j. overington	PERSON
admet-530	134	1	nat rev drug discov	PERSON
admet-530	134	2	10 (2011	DATE
admet-530	134	3	197	CARDINAL
admet-530	135	1	7	CARDINAL
admet-530	135	2	leeson	PERSON
admet-530	137	1	journal of medicinal chemistry	ORG
admet-530	137	2	2018	DATE
admet-530	138	1	8	CARDINAL
admet-530	138	2	hill	ORG
admet-530	138	3	r.j.	PERSON
admet-530	140	1	today 15 (2010	DATE
admet-530	140	2	648-655	CARDINAL
admet-530	141	1	9	CARDINAL
admet-530	141	2	k. valko	PERSON
admet-530	141	3	c. bevan	PERSON
admet-530	141	4	d. reynolds	PERSON
admet-530	141	5	69 (1997	DATE
admet-530	141	6	2022	CARDINAL
admet-530	142	1	10	CARDINAL
admet-530	142	2	d.v. green	PERSON
admet-530	142	3	c.n.	GPE
admet-530	142	4	luscombe	GPE
admet-530	142	5	a.p.	GPE
admet-530	142	6	hill.	PERSON
admet-530	144	1	today 16 (2011) 822830	DATE
admet-530	145	1	11	CARDINAL
admet-530	145	2	g. caron	PERSON
admet-530	145	3	m. vallaro	PERSON
admet-530	145	4	g. ermondi	GPE
admet-530	145	5	g.h. goetz	ORG
admet-530	145	6	l. philippe	PERSON
admet-530	145	7	m. shalaeva	PERSON
admet-530	147	1	13	CARDINAL
admet-530	147	2	2016	CARDINAL
admet-530	147	3	1100-1110	DATE
admet-530	148	1	12	CARDINAL
admet-530	150	1	130	CARDINAL
admet-530	150	2	2016	CARDINAL
admet-530	150	3	35	CARDINAL
admet-530	151	1	13	CARDINAL
admet-530	151	2	m.k. bayliss	PERSON
admet-530	151	3	j. butler	PERSON
admet-530	151	4	p.l. feldman	PERSON
admet-530	151	5	d.v. green	PERSON
admet-530	151	6	leeson	PERSON
admet-530	151	7	m.r. palovich	GPE
admet-530	151	8	a.j. taylor	PERSON
admet-530	153	1	today 21	DATE
admet-530	153	2	1719-1727	DATE
admet-530	154	1	14	CARDINAL
admet-530	154	2	c. horváth	PERSON
admet-530	154	3	w. melander	PERSON
admet-530	154	4	i. molnár	PERSON
admet-530	156	1	125	CARDINAL
admet-530	156	2	1976	DATE
admet-530	156	3	129	CARDINAL
admet-530	157	1	6(2	CARDINAL
admet-530	157	2	2018	DATE
admet-530	157	3	74	CARDINAL
admet-530	157	4	10.5599	CARDINAL
admet-530	157	5	83	CARDINAL
admet-530	158	1	15	CARDINAL
admet-530	158	2	f. lombardo	PERSON
admet-530	158	3	m.y.	ORG
admet-530	158	4	k.a. tupper	PERSON
admet-530	158	5	f. gao	PERSON
admet-530	159	1	elogdoct	PERSON
admet-530	160	1	2	CARDINAL
admet-530	161	1	journal of medicinal chemistry	ORG
admet-530	161	2	44 (2001) 24902497	DATE
admet-530	162	1	16	CARDINAL
admet-530	162	2	a. vailaya	PERSON
admet-530	162	3	c. horváth	PERSON
admet-530	164	1	101	CARDINAL
admet-530	165	1	17	CARDINAL
admet-530	165	2	k. valkó	PERSON
admet-530	165	3	l.r	DATE
admet-530	165	4	j.l.	GPE
admet-530	167	1	656	CARDINAL
admet-530	167	2	1993	DATE
admet-530	167	3	501	CARDINAL
admet-530	168	1	18	CARDINAL
admet-530	168	2	waring	ORG
admet-530	170	1	opin	PERSON
admet-530	170	2	5	CARDINAL
admet-530	170	3	2010	DATE
admet-530	170	4	235	CARDINAL
admet-530	171	1	19	CARDINAL
admet-530	171	2	c. hansch	PERSON
admet-530	171	3	j.p. bjorkroth	PERSON
admet-530	171	4	a. leo.	PERSON
admet-530	172	1	76	CARDINAL
admet-530	172	2	1987	DATE
admet-530	172	3	663	CARDINAL
admet-530	173	1	20	CARDINAL
admet-530	173	2	g.m.	PERSON
admet-530	173	3	keseru	GPE
admet-530	173	4	p.d. leeson	PERSON
admet-530	173	5	d.c. rees	PERSON
admet-530	173	6	reynolds	PERSON
admet-530	174	1	discovery	PRODUCT
admet-530	175	1	nat rev drug discov	PERSON
admet-530	175	2	13	CARDINAL
admet-530	175	3	2014	DATE
admet-530	175	4	105	CARDINAL
admet-530	176	1	21	CARDINAL
admet-530	176	2	ritchie	PERSON
admet-530	176	3	s.j. macdonald	PERSON
admet-530	177	1	discovery	PRODUCT
admet-530	178	1	journal of medicinal chemistry	ORG
admet-530	178	2	57	DATE
admet-530	178	3	2014	DATE
admet-530	178	4	7206-7215	DATE
admet-530	179	1	22	CARDINAL
admet-530	179	2	ritchie	PERSON
admet-530	179	3	s.j. macdonald	PERSON
admet-530	181	1	today 14 (2009	DATE
admet-530	181	2	1011	CARDINAL
admet-530	182	1	23	CARDINAL
admet-530	182	2	ritchie	PERSON
admet-530	182	3	s.j. macdonald	PERSON
admet-530	182	4	r.j. young	PERSON
admet-530	182	5	s.d. pickett	PERSON
admet-530	184	1	today 16 (2011	DATE
admet-530	184	2	164	CARDINAL
admet-530	185	1	24	CARDINAL
admet-530	185	2	k. valko	PERSON
admet-530	185	3	s. nunhuck	PERSON
admet-530	185	4	c. bevan	PERSON
admet-530	185	5	m.h. abraham	PERSON
admet-530	185	6	d.p. reynolds	GPE
admet-530	187	1	octanol	PERSON
admet-530	188	1	92	CARDINAL
admet-530	188	2	2003) 22362248	DATE
admet-530	189	1	25	CARDINAL
admet-530	189	2	s. ong	PERSON
admet-530	189	3	h. liu	PERSON
admet-530	189	4	x. qiu	GPE
admet-530	189	5	m. pidgeon	PERSON
admet-530	189	6	a.h. dantzig	ORG
admet-530	189	7	j. munroe	PERSON
admet-530	189	8	w.j. hornback	GPE
admet-530	189	9	j.s. kasher	PERSON
admet-530	191	1	38 (1995	DATE
admet-530	191	2	590	CARDINAL
admet-530	192	1	26	CARDINAL
admet-530	192	2	k. valko	PERSON
admet-530	192	3	c.d. bevan	PERSON
admet-530	192	4	d.p. reynolds	PERSON
admet-530	192	5	m.h. abraham	PERSON
admet-530	194	1	89	CARDINAL
admet-530	194	2	2000	DATE
admet-530	194	3	1085-1096	DATE
admet-530	195	1	27	CARDINAL
admet-530	195	2	t. vallianatou	GPE
admet-530	195	3	a. tsantili-kakoulidou	PERSON
admet-530	197	1	11	CARDINAL
admet-530	197	2	2016) 473488	DATE
admet-530	198	1	28	CARDINAL
admet-530	199	1	p. vitovič	PERSON
admet-530	200	1	kinnunen	PERSON
admet-530	202	1	4	CARDINAL
admet-530	202	2	2009	DATE
admet-530	202	3	1224	CARDINAL
admet-530	203	1	29	CARDINAL
admet-530	203	2	n. anderson	PERSON
admet-530	203	3	j. borlak	PERSON
admet-530	205	1	580	CARDINAL
admet-530	205	2	2006	DATE
admet-530	206	1	30	CARDINAL
admet-530	206	2	s. braggio	PERSON
admet-530	206	3	d. montanari	PERSON
admet-530	206	4	t. rossi	PERSON
admet-530	207	1	e. ratti	PERSON
admet-530	208	1	5	CARDINAL
admet-530	208	2	2010	DATE
admet-530	208	3	609	CARDINAL
admet-530	209	1	31	CARDINAL
admet-530	209	2	k.l.	GPE
admet-530	209	3	s.b.	PERSON
admet-530	209	4	nunhuck	GPE
admet-530	209	5	a.p. hill	GPE
admet-530	211	1	journal of pharmaceutical sciences	ORG
admet-530	211	2	100	CARDINAL
admet-530	211	3	2011	DATE
admet-530	211	4	849	CARDINAL
admet-530	212	1	32	CARDINAL
admet-530	212	2	k. valko	PERSON
admet-530	212	3	e. chiarparin	PERSON
admet-530	212	4	s. nunhuck	PERSON
admet-530	212	5	d. montanari	PERSON
admet-530	214	1	journal of pharmaceutical sciences	ORG
admet-530	214	2	101	CARDINAL
admet-530	214	3	2012	DATE
admet-530	214	4	4155-4169	DATE
admet-530	215	1	33	CARDINAL
admet-530	215	2	k.l. valko	GPE
admet-530	215	3	teague	ORG
admet-530	215	4	c. pidgeon	PERSON
admet-530	217	1	5	CARDINAL
admet-530	217	2	2017	CARDINAL
admet-530	217	3	14	CARDINAL
admet-530	218	1	s. bunnally	PERSON
admet-530	218	2	r.j. young admet &	ORG
admet-530	218	3	6(2	CARDINAL
admet-530	218	4	2018	DATE
admet-530	218	5	74-84 84	PERCENT
admet-530	218	6	34	CARDINAL
admet-530	218	7	s. teague	PERSON
admet-530	218	8	k. valko	PERSON
admet-530	219	1	discovery	PRODUCT
admet-530	220	1	european journal of pharmaceutical sciences	ORG
admet-530	220	2	110	CARDINAL
admet-530	220	3	2017	CARDINAL
admet-530	220	4	37	CARDINAL
admet-530	221	1	2018	DATE
admet-530	222	1	iapc	ORG
admet-530	222	2	zagreb	GPE
admet-530	222	3	croatia	GPE
admet-530	223	1	http://creativecommons.org/licenses/by/3.0/	ORG
admet-530	223	2	http://creativecommons.org/licenses/by/3.0/	ORG
